Histone-induced damage of a mammalian epithelium: the conductive effect. Kleine, Teri J., Amy Gladfelter, Peter N. Lewis, and Simon A. Lewis. Department of Physiology and Biophysics, University of Texas Medical Branch, 301 University Blvd., Galveston, TX, 77555-0641, Telephone Number 409-772-3397, FAX Number 409-772-3381
APStracts 2:0035C, 1995.
Human semen has been reported to be cytotoxic to rat descending colon by a mechanism involving polyamines (cationic molecules) and collagenase. In this study we report that histones, cationic proteins found in human semen, can contribute to semen's cytotoxicity. Histones H1, H4 and H5, when added to the mucosal-side of rabbit urinary bladder epithelium, were found to alter the transepithelial conductance (Gt) in a voltage-sensitive manner. When the cell interior was negative, the conductance rapidly increased and plateaued. When the cell interior was positive, the induced-conductance decreased to control values. Histone increased the Gt by increasing the apical membrane conductance rather than the tight junction conductance. The magnitude of the Gt increase was dose-dependent, and the histone-induced conductance was non -selective for sodium, potassium, and chloride. The induced conductance could be reversed by either increasing mucosal calcium concentration or by removal of histone from the mucosal solution. Prolonged exposure of the epithelium to histone was toxic as determined by the irreversible loss of transepithelial resistance. These results indicate that histone increases membrane ionic permeability, is cytotoxic, and thus may contribute to human semen's toxic effect on colonic epithelium.

Received 1 August 1994; accepted in final form 16 November 1994
APS Manuscript Number C0452-4.
Article publication pending Am. J. Physiol. (Cell Physiology).
ISSN 1080-4757 Copyright 1994 The American Physiological Society.
Published in APStracts on 27 February 1995.