Modulation of cell membrane potential in cultured vascular endothelium. Vaca, L Licea A & Possani Ld. Department of Molecular Physiology and Biophysics, Baylor College of Medicine, Houston, Texas 77030 and Departamento de Bioenergetica y Biomembranas, Instituto de Fisiologia Celular, Uiversidad Nacional Autonoma de Mexico, Apartado Postal 70-600, Mexico D. F. 04510, Department of Molecular Recognition and Structural Biology, Instituto de Biotecnologia, Universidad Nacional Autonoma de M[acute]exico. Apartado Postal 510-3,, Cuernavaca, Morelos 62271, M[acute]exico
APStracts 2:0357C, 1995.
The present study explores the role of different ionic conductances in the regulation of membrane potential under resting conditions and after bradykinin or thapsigargin stimulation of cultured bovine aortic endothelial cells (BAEC). Under resting conditions the cell membrane potential observed was -62 5 mV. The main conductance under these conditions is an inwardly rectifying potassium channel (IRK). Application of 50 nM bradykinin (Bk) induced a transient hyperpolarization to -87 4 mV followed by a sustained depolarization to -35 5 mV. The transient hyperpolarization was eliminated by 1 [mu]M noxiustoxin (NTX), a blocker of calcium-activated potassium channels (KCa). The sustained depolarization induced by Bk was prevented by incubating the cells with the calcium channel blocker lanthanum (La3+). Thapsigargin (TG) evoked a similar response in membrane potential with the exception that the onset of the hyperpolarization was slower compared to Bk. The results presented here indicate that the cell resting potential is maintained at -62 2 mV by the IRK. Bk or TG stimulation induces a transient hyperpolarization of approximately -20 mV produced by activation of a KCa channel. This hyperpolarization is followed by a sustained depolarization produced by activation of a calcium selective channel sensitive to La3+.

Received 18 August 1995; accepted in final form 20 September
1995.
APS Manuscript Number C514-5.
Article publication pending Am. J. Physiol. (Cell Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 6 November 95