Recovery from nmda-induced intracellular acidification in cortical neurons is delayed and dependent on extracellular bicarbonate. Canzoniero, L. M. T., S. L. Sensi, and D. W. Choi. Center for the Study of Nervous System Injury, and Department of Neurology, Washington University School of Medicine, St. Louis, MO 63110
APStracts 2:0331C, 1995.
A thirty second exposure to N-methyl-D-aspartate (NMDA) produced a dose-dependent and long-lasting (10-20 min) reduction in intracellular pH in cultured cortical neurons, detected by the fluorescent dye 2,7' bis-carboxyethyl 5,6 carboxy-fluorescein (BCECF). This intracellular acidification could be blocked by addition of the NMDA antagonist, D(-)-2-amino-5-phosphonovalerate (D -APV), or by removal of extracellular Ca2+. Removal of extracellular HCO3- markedly impaired recovery from NMDA-induced intracellular acidification. Recovery was also impaired when 4,4' -diisothiocyanostilbene-2,2'-disulphonic acid (DIDS) or 4-acetamido -4'-isothiocyanato-stilbene-2,2'-disulfonic acid (SITS), inhibitors of HCO3- transport, were added to the cultures immediately after NMDA exposure. In contrast, the Na+ - H+ exchange blocker, 5-(N-ethyl-N -isopropyl)amiloride (EIPA) did not affect pH recovery. Removal of extracellular Cl- ions partially prevented pH recovery after NMDA stimulation. In addition, extracellular HCO3- increased intracellular Na+ after NMDA exposure, consistent with HCO3- activation of a Na+ -dependent exchanger. These results demonstrate that stimulation of cortical neuronal NMDA receptors is followed by long-lasting intracellular acidification, and that the presence of extracellular HCO3- is important in the subsequent recovery of normal intracellular pH, likely acting at least in part via the Na+ -dependent Cl--HCO3- exchanger.

Received 10 November 1994; accepted in final form 5 September
1995.
APS Manuscript Number C666-4.
Article publication pending Am. J. Physiol. (Cell Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 23 September 1995.