Glycine minimizes reperfusion injury in a low-flow, reflow liver perfusion model in the rat. Zhong, Zhi, Shannon Jones, and Ronald G. Thurman. Laboratory of Hepatobiology and Toxicology, Department of Pharmacology, University of North Carolina at Chapel Hill, Chapel Hill, NC 27514
APStracts 2:0154G, 1995.
This study investigated the effects of glycine on reperfusion injury in a low-flow, reflow liver perfusion model. With this protocol, livers were perfused at low flow rates around 1 ml/g/min for 75 min, which caused cells in pericentral regions of the liver lobule to become anoxic because of insufficient delivery of oxygen. When normal flow rates (about 4 ml/g/min) were restored for 40 min, an oxygen -dependent reperfusion injury occurred. Upon reflow, lactate dehydrogenase (LDH), a cytosolic enzyme, and malondialdehyde (MDA), an end product of lipid peroxidation, were released into the effluent perfusate. LDH increased from basal levels of about 1 to 35 IU/g/h in livers from control rats. Glycine (0.06-2.00 mM) minimized enzyme release in a dose-dependent manner (half-maximal decrease =133 [mu]M), with maximal values only reaching 5 IU/g/h when glycine was increased to 2 mM. Reflow for 40 minutes following 75 minutes of low -flow hypoxia caused death in about 30% of previously anoxic parenchymal cells in pericentral regions; however, infusion of glycine (2 mM) decreased cell death to less than 10%. Strychnine (1 mM), which was found to mimic the cytoprotective effect of glycine in proximal renal tubules, also reduced LDH release to 11 IU/g/h in this study. Bile was released at rates of around 42 [mu]l/g/h in livers from control rats but values were not altered significantly by glycine. Maximal MDA production during reperfusion decreased by 35% with 0.6 mM of glycine. Trypan blue distribution time, an indicator of hepatic microcirculation, was reduced significantly by glycine at 5 and 40 minutes after reflow, but changes were about 2-fold greater at later than earlier time points (half-maximal decrease = 225 [mu]M). Time for oxygen to reach steady state upon reflow was reduced by glycine in a dose-dependent manner, and the rates of entry and exit of a dye confined to vascular space (fluorescein-dextran) were increased 2 to 3-fold by glycine, respectively. Taken together, these data indicate that a reperfusion injury, which occurs in previously hypoxic pericentral regions of the liver upon reintroduction of oxygen, is minimized by glycine, possibly by action on a glycine -sensitive anion channel to improve microcirculation during the reperfusion period.

Received 18 January 1995; accepted in final form 17 July 1995.
APS Manuscript Number G23-5.
Article publication pending Am. J. Physiol. (Gastrointest. Liver
Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 10 August 1995.