Microvascular dysfunction induced by nonsteroidal anti-inflammatory drugs: role of leukocytes. Kurose, Iwao, Robert Wolf, Masayuki Miyasaka, Donald C. Anderson, and D. Neil Granger. Departments of Physiology and Medicine, Center of Excellence in Arthritis and Rheumatology, Louisiana State University Medical Center, Shreveport, LA, 71130-3932, Department of Bioregulation, Osaka University Medical School, Discovery Research, UpJohn Laboratories, Kalamazoo, MI
APStracts 2:0170G, 1995.
The objectives of this study were to determine whether 1) the leukocyte-endothelial cell adhesion observed in venules exposed to nonsteroidal anti-inflammatory drugs (NSAIDs) is accompanied by enhanced albumin extravasation, and 2) leukocytes mediate this endothelial cell barrier dysfunction. Intravital video microscopy was used to monitor leukocyte-endothelial cell adhesion and the leakage of FITC- labelled albumin in rat mesenteric venules exposed to either indomethacin or aspirin. Both NSAIDs induced the recruitment of adherent and emigrated leukocytes, with temporally related increases in albumin leakage. Agents that effectively decreased or prevented the NSAID- induced leukocyte adherence/emigration (leukotriene B4 receptor antagonist or adhesion molecule-specific monoclonal antibodies) also blocked the corresponding albumin leakage response. These findings indicate that adherent and/or emigrating leukocytes mediate the early endothelial cell barrier dysfunction elicited by NSAIDs.

Received 27 April 1995; accepted in final form 3 August 1995.
APS Manuscript Number G177-5.
Article publication pending Am. J. Physiol. (Gastrointest. Liver
Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 24 August 1995.