Linkage of [ca2+]i in single isolated d-cells to somatostatin secretion induced by cholecystokinin. Delvalle, J., J. Wakasugi, H. Takeda, and T. Yamada. Departments of Internal Medicine and Physiology, The University of Michigan Medical Center, Ann Arbor, Michigan 48109
APStracts 2:0243G, 1995.
The Ca2+/inositol phospholipid signaling cascade has been implicated in the mechanism by which cholecystokinin (CCK) stimulates gastric somatostatin release, but a direct linkage between intracellular events in gastric D-cells and somatostatin secretion has not been established. To address this problem we developed a method for correlating somatostatin release with the measurement of [Ca2+]i in isolated D-cells. Resting [Ca2+]i in single D-cells was 100 +/- 5.7 nM (mean +/- SE, n = 41) and CCK induced a rise in [Ca2+]i in a dose dependent fashion, producing a maximal stimulatory effect (243 +/- 15% of control, n = 12) at a peptide concentration of 2 x 10-8M. The CCK mediated increase in [Ca2+]i was biphasic, with a rapid, initial transient elevation, followed by a sustained plateau. The rise in [Ca2+]i was accompanied by a concomitant increase in release of somatostatin like immunoreactivity (SLI). Removal of extracellular Ca2+ had no effect on the initial transient elevation in [Ca2+]i induced by CCK but abolished both the sustained plateau in [Ca2+]i and the release of SLI. The selective CCK antagonist L-364,718 (10 -7M) inhibited the effects of CCK on both [Ca2+]i and SLI release. The nonspecific Ca2+ channel blocker NiCl2 (10-3M) and the L-type calcium channel blocker, nifedipine, inhibited the sustained rise in [Ca2+]i and the release of SLI, but left unaltered the initial transient increase in [Ca2+]i. These results indicate that CCK stimulated release of SLI from D-cells in the gastric fundus is linked to influx of extracellular Ca2+ via L-type Ca2+ channels.

Received 25 September 1995; accepted in final form 7 November
1995.
APS Manuscript Number G419-5.
Article publication pending Am. J. Physiol. (Gastrointest. Liver
Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 8 December 95