In vivo production of nitric oxide correlates with n-methyl-d- aspartate-induced cerebral hyperemia in newborn sheep. Northington, Frances J., Joseph R. Tobin, Raymond C. Koehler, and Richard J. Traystman. The Johns Hopkins Medical Institutions, Departments of Pediatrics and Anesthesiology/Critical Care Medicine, Baltimore, Maryland 21287
APStracts 2:0045H, 1995.
Stimulation of N-methyl-D-aspartate (NMDA) receptors in brain increases nitric oxide production in vitro. We tested the hypothesis that nitric oxide participates in the increase in local cerebral blood flow (CBF) caused by infusion of NMDA in anesthetized newborn sheep. We used the combined hydrogen clearance and microdialysis technique for simultaneous measurement of local CBF, infusion of drugs, and measurement of interstitial levels of [14C]-L -citrulline in the parietal cortex. Release of [14C]-L -citrulline into the dialysate during continuous infusion of [14C]-L-arginine was used as a marker of nitric oxide production in vivo. Citrulline recovery and CBF were measured hourly during a 4 hour infusion of cerebrospinal fluid containing either 1) no additional drugs, 2) 1 mM NMDA, 3) 1mM NG-nitro-L-arginine methyl ester (L-NAME, a nitric oxide synthase inhibitor), 4) 1 mM NMDA+1mM L-NAME, 5) 0.1 mM 2-chloroadenosine (adenosine receptor agonist)and 6) 0.1 mM 2-chloroadenosine +1mM L-NAME. At 240 minutes of perfusion, CBF (ml_min-1_100g-1); (mean +/- SE) was: control 52+/-3, NMDA 116+/-11, L -NAME 32+/-5, NMDA+L-NAME 40+/-4, 2-chloroadenosine 201+/-63 and 2 -chloroadenosine+L-NAME 129+/-18. Citrulline recovery (femtomoles/min) at 240 minutes of perfusion was: control 38+/-12, NMDA 149+/-21, L-NAME 9+/-1, NMDA+L-NAME 39+/-5, 2-chloroadenosine 13+/-5, 2-chloroadenosine + L -NAME 17+/-1. Infusion of NMDA increased CBF and [14C]-L -citrulline release and these increases were inhibited by addition of L-NAME to the dialysate. In contrast, the cerebral vasodilator, 2 -chloroadenosine, with or without L-NAME increased CBF without an increase in [14C]-L-citrulline release, thereby demonstrating that the effect of L-NAME to block NMDA-mediated increases in CBF was specific and not due to generalized vasoparalysis. These results demonstrate that the local increase in CBF caused by stimulation of cortical NMDA receptors is dependent on production of nitric oxide. This study also demonstrates that microdialysate-measured conversion of [14C]-L-arginine to [14C]-L-citrulline is potentially useful as a marker of nitric oxide production in vivo.

Received 12 April 1994; accepted in final form 7 February 1995.
APS Manuscript Number H322-4.
Article publication pending Am. J. Physiol. (Heart Circ. Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 24 February 1995.