Cardiac responses to induced lactate oxidation: nmr analysis of metabolic equilibria. Lewandowski, E. Douglas, Lisa A. Damico, Lawrence T. White, and Xin Yu. NMR Center, Department of Radiology, Massachusetts General Hospital, Harvard Medical School, Boston, MA
APStracts 2:0048H, 1995.
The role of lactate, as a source of pyruvate oxidation in supporting cardiac work, energetics, and formation of oxidative metabolites, was examined in normal myocardium. 13C and 31P NMR spectra were acquired from isolated rabbit hearts supplied 2.5 mM [3-13C] lactate or [3-13C] pyruvate with or without stimulation of pyruvate dehydrogenase (PDH) by dichloroacetate (DCA). Similar workloads determined by rate pressure products were noted with pyruvate (21700+2400; Mean+SE) and lactate (18970+1510). Oxygen consumption was similar in all four groups with means between 19.0 - 22.2 [mu]mol/min/g dry weight (SE= 1.6-2.0) as was the ratio of phosphocreatine to ATP with means between 1.8 - 2.1 (SE = 0.1 - 0.6). Intracellular pH, determined from 31P NMR spectra, was essentially the same with pyruvate (7.06 +/- 0.02) and lactate (7.05 +/- 0.04). 13C enrichment of glutamate was higher with lactate (92%) than pyruvate (70%). Pyruvate plus DCA induced no change in glutamate content at 9 -10 [mu]mol/g, but 13C-enrichment increased to 83%, while lactate plus DCA maintained enrichment at 90%. Levels of [alpha]-ketoglutarate were lower with lactate (1.81 [mu]mol/g) than with pyruvate (2.36 [mu]mol/g). Lactate plus DCA elevated glutamate by 60% with a proportional increase in [alpha]-ketoglutarate. Thus, the balance between glutamate and [alpha]-ketoglutarate was affected by substrate supply only and not by PDH activation. The results suggest that the equilibrium between [alpha] -ketoglutarate and glutamate is sensitive to cytosolic redox state, an important consideration for 13C NMR analyses that rely on glutamate. In conclusion, lactate and pyruvate are able to support similar function and energetics through differences in the balance of oxidative, intermediary metabolites.

Received 17 October 1994; accepted in final form 31 January 1995.
APS Manuscript Number H932-4.
Article publication pending Am. J. Physiol. (Heart Circ. Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 24 February 1995.