Constitutive nitric oxide synthase protein and mrna levels are elevated in cultured human and bovine endothelial cells exposed to fluid shear stress. Ranjan, Vibhu, Zeshuai Xiao, Scott L. Diamond. Bioengineering Laboratory, Department of Chemical Engineering, The State University of New York, Buffalo, NY 14260, Tel (716) 645-2911 ext. 2205, Fax (716) 645-3822
APStracts 2:0064H, 1995.
Flow induced activation of nitric oxide synthase (NOS) in endothelial cells causes vasodilation due to a burst in NO production, particularly when prevailing flows change acutely. The role of chronic fluid shear stress exposures on endothelial constitutive nitric oxide synthase (cNOS) levels may also have an important role in vessel diameter control. To test the role of sustained flow exposures, we subjected primary human umbilical vein endothelial cells (HUVEC) or bovine aortic endothelial cells (BAEC, passage 2-14) to steady laminar shear stress using a parallel-plate flow apparatus. In both endothelial cell types, the intracellular level of cNOS was elevated within 3 hr of flow exposure at 25 dynes/cm2 and remained elevated at 6 and 12 hours of flow exposure, compared to stationary controls, as indicated by digital immunofluorescence microscopy. Shear stress exposure for 6 hr caused a 2.2 +/- 0.3 and 2.8 +/- 0.3 -fold elevation of cNOS proteins levels in BAEC (n = 3, p<0.01) and HUVEC (n = 3, p<0.01), respectively, in the presence or absence of 1 [mu]M dexamethasone. Dexamethasone suppresses induction of the inducible NOS gene, indicating that constitutive NOS was elevated by fluid shear stress. Flow exposure at 4 dynes/cm2 caused no enhancement of cNOS levels in either cell type. The flow induction of the cNOS protein levels was not blocked by preincubation of BAEC with 100 to 400 [mu]M of NG-nitro-L-arginine methyl ester, indicating that a positive feedback loop for flow induced NO (or cGMP) was not involved in the elevation of cNOS levels. Also the protein kinase C inhibitor, H7 (10 [mu]M) had no effect on induction of NOS protein in BAEC exposed to 25 dynes/cm2. The cNOS mRNA levels were found to be elevated by 2 to 3-fold in BAEC after 6 or 12 hours of flow exposure at either 4 or 25 dynes/cm2, and this induction of NOS mRNA occurred in the presence of dexamethasone. The rapid and sustained elevation of endothelial NOS levels by chronic flow exposure in coordination with the sustained suppression of endothelin-1 gene expression by arterial levels of shear stress may provide a mechanism at the level of gene expression for chronic regulation of vessel diameter by endothelial response to prevailing blood flow.

Received 18 November 1994; accepted in final form 15 February
1995.
APS Manuscript Number H1031-4.
Article publication pending Am. J. Physiol. (Heart Circ. Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 10 March 1995.