Effects of glucose deprivation on NMDA-induced current and intracellular Ca 2+ in rat substantia nigra neurons. Nakashima, Yasunori, Hitoshi Ishibashi, Nobutoshi Harata, and Norio Akaike. Department of Anesthesiology and Critical Care Medicine, and Department of Physiology, Faculty of Medicine, Kyushu University, 812-82, Japan .
APStracts 2:0288N, 1995.
SUMMARY AND CONCLUSIONS
1. The effects of glucose deprivation on N -methyl- D -aspartate (NMDA)- induced current (I NMDA ) and the intracellular free Ca 2+ concentration ([Ca 2+ ] i ) in the acutely dissociated rat substantia nigra neurons were investigated using the nystatin-perforated patch-clamp technique under voltage-clamp and the microfluometry with a fluorescent probe, Indo-1. 2. Application of NMDA induced a peak and a successive steady-state inward currents, and an outward current immediately after washout at a holding potential of -40 mV. The amplitudes of the three current components of I NMDA were increased by increasing the concentrations of NMDA with the half-maximum concentration (EC 50 ) of 1.1 [lambda] 10 -4 , 1.2 [lambda] 10 -4 and 1.6 [lambda] 10 -4 M, respectively. 3. The reversal potentials of the peak inward and outward currents were -4 +/- 3 and -76 +/- 2 mV, respectively. The latter was close to the theoretical K + equilibrium potential (-82 mV). 4. The outward current was potentiated by increase in extracellular Ca 2+ concentration and was blocked by Cs + -internal solution, suppressed by 5 [lambda] 10 -3 M tetraethylammonium chloride and 10 -7 M charybdotoxin, indicating that it was Ca 2+ -activated K + current (I K(Ca) ). 5. Application of NMDA concentration-dependently increased [Ca 2+ ] i with EC 50 of 3.9 [lambda] 10 -5 M. 6. Deprivation of glucose from the external solution induced a slowly developing outward current and increased the basal level of [Ca 2+ ] i . It also prolonged the NMDA-induced outward current without affecting the peak inward current, and prolonged the NMDA-induced increase in [Ca 2+ ] i without changing the peak [Ca 2+ ] i . 7. These findings suggest that the deprivation of glucose did not affect the NMDA-induced influx of Ca 2+ into the cells, but it inhibited Ca 2+ clearance by affecting the efflux of Ca 2+ to the extracellular space, re-uptake into the intracellular Ca 2+ stores, and/or active extrusion from intracellular stores.

Received 13 April 1995; accepted in final form 12 September 1995.
APS Manuscript Number J244-5.
Article publication pending J. Neurophysiol.
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 31 October 95