Studies of renal injury i. gentamicin toxicity and the expression of genes encoding basolateral transporters of rat renal proximal tubules. Dominguez, Jesus H., Calvin C. Hale, and Mona Qulali. Department of Medicine, Department of Physiology and Biophysics, Indiana University Medical Center and Veterans Administration Medical Center, Indianapolis, Indiana 46202; and Department of Veterinarian Medical Sciences, John M. Dalton Research Center, University of Missouri, Columbia, Missouri 65211
APStracts 2:0129F, 1995.
Gentamicin nephrotoxicity may arise in part from alterations in the expression of genes critical for renal proximal tubule metabolism. We tested the hypothesis that gentamicin suppressed the gene expression of the Na+/Ca2+ exchanger (NaCaX), glucose transporter 1 (GLUT1) and 1 subunit of Na+/K+ ATPase (1 NKA) in renal tubules. The products of these genes mediate Na+-dependent Ca2+ efflux, glucose efflux and influx, and ATP-dependent Na+ efflux across tubular basolateral membranes, respectively. After 10 days of gentamicin intoxication (40 mg/kg/twice daily, I.P.), levels of mRNAs encoding NaCaX and the cognate protein declined. GLUT1 mRNA levels increased, although GLUT1 protein levels were also reduced. Moreover, whereas [alpha]1 NKA mRNA levels remained unchanged, [alpha]1 NKA protein levels were also reduced. We suggest that the higher GLUT1 mRNA level is part of the stress response to tubular injury. However, regardless of the mRNA level, the most consistent effect of gentamicin was reduction of specific protein levels. We propose that failure to translate high levels of mRNA into proportionally high levels of protein, as in the case of GLUT1, may attenuate the expression of stress response gene products; and thus diminsh the possibility of recovery in gentamicin intoxication.

Received 18 October 1994; accepted in final form 17 July 1995.
APS Manuscript Number F376-4.
Article publication pending Am. J. Physiol. (Renal Fluid Electrolyte
Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 10 August 1995.