Hypertonic nacl enhances adenosine release and hormonal camp production in mouse thick ascending limb. Baudouin-Legros, Maryvonne, Abdallah Badou, Marc Paulais, Mich[grave]ele Hammet, and Jacques Teulon. INSERM U323, Facult[acute]e de M[acute]edecine Necker-Enfants Malades, 156 rue de Vaugirard, 75015 PARIS FRANCE, Phone: 1 40 61 56 22; Fax: 1 40 61 55 91
APStracts 2:0027F, 1995.
Cyclic AMP (cAMP) accumulated in the presence of adenosine was measured in medullary portions of mouse thick ascending limbs of Henle's loop (mTAL) suspended either in classical extracellular buffer, or in the presence of added NaCl. Under control conditions (NaCl:140 mmol/l), adenosine (<10-5 mol/l) and CHA (N6 -cyclohexyladenosine, an A1 adenosine receptor agonist) inhibit the cAMP accumulation induced by arginine-vasopressin (AVP). On the other hand, high concentrations of adenosine and CGS21680 (2 -[p(carboxyethyl)phenethylamino]-5'-N-ethylcarboxamidoadenosine, an A2 adenosine receptor agonist) stimulate cAMP formation. Addition of NaCl (+ 300 mmol/l) to extracellular buffer stimulates the release of endogenous adenosine. It also enhances A2R-induced cAMP accumulation but suppresses A1R-mediated inhibition of adenylyl cyclase. This hypertonic NaCl medium also potentiates the stimulatory action of arginine-vasopressin on adenylyl cyclase. The modifications of tubular responses to both AVP and A1 and A2 agonists brought about by hypertonic NaCl were all inhibited by adenosine deaminase, thereby demonstrating the involvement of endogenous adenosine. Adenosine, the release and the effects of which are modulated by hypertonic NaCl, thus appears to act as an endogenous physiological modulator of kidney medulla function.

Received 28 July 1994; accepted in final form 21 February 1995.
APS Manuscript Number F264-4.
Article publication pending Am. J. Physiol. (Renal Fluid Electrolyte
Physiology).
ISSN 1080-4757 Copyright 1995 The American Physiological Society.
Published in APStracts on 10 March 1995.