Roles of cytoplasmic ca2& and intracellular ca2& stores in induction and suppression of apoptosis in s49 cells. Bian, Xiaopeng, Francis M. Hughes, Jr., Yi Huang, John A. Cidlowski, James W. Putney, Jr. Laboratory of Cellular and Molecular Pharmacology, National Institute of Environmental Health Sciences, National Institutes of Health, Research Triangle Park, North Carolina 27709
APStracts 3:0368C, 1996.
The Ca2&-ATPase inhibitors, thapsigargin and cyclopiazonic acid, depleted intracellular Ca2& stores, induced large increases in [Ca2&]i, and caused apoptosis in S49 cells. Removal of extracellular Ca2& augmented apoptosis due to thapsigargin, indicating that depletion of Ca2& from intracellular stores is responsible for apoptosis with this agent. Overexpression of the apoptosis suppressor, Bcl-2, inhibited apoptosis due to thapsigargin, but did not affect thapsigargin-induced Ca2& signalling. Dexamethasone induced apoptosis, diminished the size of the endoplasmic reticulum Ca2& pool, and caused a small elevation of intracellular Ca2&. However, this elevation was not due to Ca2& influx because the increase was similar in the presence or absence of Ca2& in the medium. Furthermore, in contrast to the results with thapsigargin, apoptosis due to dexamethasone was unchanged in a Ca2&-free medium. These results indicate that depletion of Ca2& stores initiates a pathway leading to apoptosis. Elevations in cytoplasmic Ca2& appears to play a lesser role than previously thought in the actions of Bcl-2 and glucocorticoids.

Received 6 June 1996; accepted in final form 19 November 1996.
APS Manuscript Number C317-6.
Article publication pending Am. J. Physiol. (Cell Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 31 December 1996