Extracellular atp modulates [ca2+]i in retinoic acid-treated embryonic chondrocytes. Hung, Clark T., Fred D. Allen, Kyle D. Mansfield, and Irving M. Shapiro. Center for Biomedical Engineering, Columbia University, New York, NY 10032, Dept. of Bioengineering, School of Engineering and Applied Sciences, Univ. of Pennsylvania, Philadelphia, PA 19104-6392, Dept. of Biochemistry, School of Dental Medicine, Univ. of Pennsylvania, Philadelphia, PA 19104-6003
APStracts 3:0399C, 1996.
Treated with low doses of retinoic acid (RA), cephalic chondrocytes of the chick embryonic sternum mature and express phenotypic characteristics of post-mitotic hypertrophic cells. In concert with these maturation-dependent changes, cells release adenine nucleotides into the culture medium. To ascertain if these compounds modulate chondrocyte function, we challenged chondrocytes with nucleotides and measured one determinant of the signal transduction pathway, [Ca2+]i. In the presence of micromolar concentrations of ATP, there was a dose dependent elevation in chondrocyte [Ca2+]i; ADP caused a small but significant rise in the peak [Ca2+]i response. We found that the change in the [Ca2+]i response is linked to retinoid-dependent maturation of chondrocytes. Thus, the [Ca2+]i rise was dependent on the RA concentration and treatment time. Immature caudal chondrocytes, cells that were not affected by RA, were used as control cells for this study. When treated with ATP, these cells did not exhibit a [Ca2+]i response. Although the purinergic subtype receptor was not characterized, the observation that cells responded to ATP and ADP, but were refractory to AMP and adenosine suggested that P2 receptors were expressed by chondrocytes. Since during the same culture period, chondrocytes exhibited many of the unique characteristics of the terminally differentiated cell, the acquisition of purinergic receptors represents a new feature associated with expression of the mature phenotype. Finally, to ascertain if the ATP-dependent response was due to release of Ca2+ from intracellular stores, cells were treated with thapsigargin. As this compound significantly reduced the [Ca2+]i signal, we concluded that the ATP response is mediated by release of cations from the endoplasmic reticulum.

Received 31 July 1996; accepted in final form 4 December 1996.
APS Manuscript Number C428-6.
Article publication pending Am. J. Physiol. (Cell Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 31 December 1996