Human monocytes lose 5-lipoxygenase and its activating protein as they mature into monocyte-derived macrophages in vitro. Ring, William L., Carl A. Riddick, Joseph R. Baker, Dominic A. Munafo, and Timothy D. Bigby. Department of Medicine, University of California, San Diego and Department of Veteran Affairs Medical Center, San Diego, California 92161
APStracts 3:0054C, 1996.
Previous studies in mononuclear phagocytes have shown that macrophages have substantially greater 5-lipoxygenase activity than monocytes and that this is associated with greater amounts of 5-lipoxygenase and its activating protein (FLAP). The aim of this study was to examine the effect of mononuclear phagocyte maturation in vitro on 5 -lipoxygenase expression. At baseline, monocytes had significant 5 -lipoxygenase activity, but then lost all detectable 5-lipoxygenase activity over seven days. Immunoblot and Northern blot analysis revealed that immunoreactive protein and mRNA for both 5-lipoxygenase and FLAP were significantly decreased over time. These studies demonstrate that in vitro differentiation of monocytes into a macrophage phenotype is not accompanied by the enhanced expression of 5-lipoxygenase and FLAP seen in macrophages derived from in vivo sources. In fact, baseline expression of 5-lipoxygenase and FLAP by monocytes is lost in vitro. These studies have clear implications for the use of cultured monocytes as a model of macrophages, and they also further our understanding of the regulation of the 5 -lipoxygenase pathway.

Received 11 December 1995; accepted in final form 26 January
1996.
APS Manuscript Number C741-5.
Article publication pending Am. J. Physiol. (Cell Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 14 February 96