Bovine adrenal endothelial cells express nucleoside transporters non-regulated by protein kinases a and c. Sen, R. P., Sobrev[acute]ia, L., Delicado, E. G., Yudilevich, D. and Miras-Portugal M. T. DEPARTMENT OF BIOCHEMISTRY. FACULTAD DE VETERINARIA. UNIVERSIDAD COMPLUTENSE. 28040 MADRID. SPAIN, DEPARTMENT OF PHYSIOLOGY, AND BIOPHYSICS, FACULTAD DE MEDICINA. UNIVERSIDAD DE CHILE. P. O. BOX 70005 SANTIAGO. CHILE.
APStracts 3:0028C, 1996.
The present investigation characterizes the nucleoside transporters in bovine adrenomedullary endothelial cells (BAMEC) and their possible regulation by the action of protein kinases A and C in order to establish comparisons with the nucleoside transport system in chromaffin cells. The nucleoside transport proved to be a NBTI -sensitive-facilitated diffusion system with high affinity for adenosine. These endothelial cells had a high density of nucleoside transporters (660,000 +/- 130,000 transporters/cell), measured by NBTI binding, and the efficiency was close to 2 molecules of adenosine internalized/transporter/second. The stimulation of the cells with bradykinin and Ap4A, which raise the intracellular Ca2+ concentration, did not modulate the adenosine transport. When the cells were stimulated with signals coupled to cAMP intracellular production, such as noradrenaline and isoproterenol, the adenosine transport was not modified. Futhermore, the treatment of the cells with direct activators of both protein kinases A and C had no effect on adenosine transport, in contrast to that reported in chromaffin cells.

Received 25 July 1995; accepted in final form 19 January 1996.
APS Manuscript Number C456-5.
Article publication pending Am. J. Physiol. (Cell Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 25 January 96