Effects of extracellular atp on ion transport and intracellular ca2+ in mongolian gerbil middle ear epithelium. Furukawa, Masayuki, Katsuhisa Ikeda, Mutsuo Yamaya, Takeshi Oshima, Hidetada Sasaki and Tomonori Takasaka. Departments of Otorhinolaryngology and Geriatric Medicine, Tohoku University School of Medicine, Sendai, Japan
APStracts 3:0356C, 1996.
The present study investigates the effects of ATP on ion transport and Ca2+ mobilization in primary cultures of gerbil middle ear epithelium. Extracellular ATP and other nucleotides elicited a transient increase in Isc in a dose-dependent manner. The rank order of potency in Isc responses corresponded with the sequence of the P2u purinergic receptor when applied to the mucosal or the basolateral side. Extracellular ATP induced a rise in the intracellular Ca2+ concentration ([Ca2+]i) in a dose-dependent manner. A similar rank order of potency in the ATP-induced increases in [Ca2+]i was observed. The time courses of the [Ca2+]i responses induced by ATP closely paralleled those of the Isc responses. 1,2-Bis-(o -aminophenoxy)ethane N,N,N,,N,-tetraacetic acid-acetoxymethyl ester greatly reduced the increase in both the Isc and [Ca2+]i responses to ATP. Diphenylamine-2-carboxylate, 4,4,-diisothiocyanostilbene-2,2, -disulfonic acid, quinidine, and Ba2+ significantly blocked the ATP -stimulated Isc. Glybenclamide had no effect on the ATP-stimulated Isc. These results are consistent with the hypothesis that extracellular ATP and other nucleotides induce Cl- secretion across the apical membrane in cultured gerbil middle ear epithelium by activation of the apical Cl- channels via multiple modes of regulation.

Received 23 July 1996; accepted in final form 8 October 1996.
APS Manuscript Number C408-6.
Article publication pending Am. J. Physiol. (Cell Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 13 November 1996