Prevention of hyperglycemia in the zucker diabetic fatty rat by treatment with metformin or troglitazone. Sreenan, Seamus, Jeppe Sturis, William Pugh, Charles F. Burant, and Kenneth S. Polonsky,. Department of Medicine The University of Chicago and Pritzker School of Medicine, Chicago, Illinois, 60637
APStracts 3:0129E, 1996.
To determine if metformin or troglitazone can delay the onset of diabetes in the Zucker diabetic fatty (ZDF) rat, lean control, fatty and ZDF rats received metformin, troglitazone or no treatment from age 6 to 12 weeks. Glucose, insulin, triglyceride (TG) and free fatty acid (FFA) levels and glucose stimulated insulin secretion by the perfused pancreas were measured. Metformin-treated rats gained significantly less weight. Both drugs prevented hyperglycemia by 12 weeks in diabetic rats and significantly reduced TG and FFA. Insulin secretion at low glucose was elevated in untreated fatty and diabetic animals and the increment in diabetic animals produced by glucose perfusion was attenuated compared to lean and fatty rats. Both drugs reduced basal insulin secretion in fatty and diabetic rats and improved glucose responsiveness in diabetic rats. Metformin and troglitazone delay onset of diabetes in the ZDF rat. The significantly improved insulin secretory response of the pancreas undoubtedly contributes to the improved glucose tolerance.

Received 23 October 1995; accepted in final form 12 June 1996.
APS Manuscript Number E509-5.
Article publication pending Am. J. Physiol. (Endocrinol. Metab.).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 25 July 1996