Carbachol but not forskolin can increase mucosal to serosal transport of intact protein in rat ileum in vitro. Bijlsma, Pieter B., Amanda J. Kiliaan, Greet Scholten, Martine Heyman, Jack A. Groot, and Jan A. J. M. Taminiau. Dept. Pediatr. Gastroenterology and Nutrition, Acad. Medical Centre, 1105 AZ Amsterdam and Dept. Exp. Zoology. University of Amsterdam. 1098 SM Amsterdam. The Netherlands. INSERM U 290, H[circumflex]opital St. Lazare, Paris, France
APStracts 3:0095G, 1996.
The effects of the secretagogues forskolin and carbachol on protein uptake in isolated ileum of rats were studied. The mucosa to serosa transport of horseradish peroxidase (HRP, MW 40 kD) was measured in Ussing chambers, and afterwards tissues were processed for electron microscopy. In the absence of secretagogues, the flux of enzymatically active HRP was 5 pmoles/cm2.h at a mucosal concentration of 10 [mu]M. Electron micrographs showed vesicles filled with active HRP in enterocytes but no HRP-activity in intercellular spaces. Forskolin decreased HRP-activity in the cells. Carbachol increased the amount of HRP-filled vesicles in enterocytes and induced HRP-filling in some intercellular spaces and tight junctions in the upper parts of the villi. The transepithelial flux of intact HRP increased more than 2.5 fold. This effect was suppressed by atropine. We conclude that cholinergic activation can increase the uptake of intact protein via endocytosis and the trans -epithelial passage by the induction of a diffusional paracellular pathway. We speculate that the increased transport of intact protein through the intestinal barrier may influence immunological sensitization to food-allergens.

Received 24 June 1995; accepted in final form 11 March 1996.
APS Manuscript Number G273-5.
Article publication pending Am. J. Physiol. (Gastrointest. Liver
Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 8 May 96