Protection of reoxygenated cardiomyocytes against osmotic fragility by no donors. Schl[umlaut]uter, K. D., G. Jakob, M. Ruiz-Meana, D. Garcia-Dorado, H. M. Piper. Physiologisches Institut, Justus-Liebig-Universit[umlaut]at Gie[beta]en, Aulweg 129, D-35392 Gie[beta]en, Germany; Servico de Cardiologia, Hospital General Universitario Vall d Hebron, Paseo Vall d Hebron 119-129, Barcelona 08035, Spain
APStracts 3:0048H, 1996.
In ischemic-reperfused myocardium, myocardial cells are jeopardized not only by reoxygenation-induced hypercontracture but also by the development of a transsarcolemmal osmotic gradient. Here, the question was addressed whether osmotic fragility of cardiomyocytes can be reduced by interventions during reoxygenation. Isolated ventricular cardiomyocytes (from adult rats), exposed to 120 min hypoxia and subsequent reoxygenation, were used as model. Upon reoxygenation medium osmolality was reduced from 270 mOsm to 80 mOsm. Loss of sarcolemmal integrity was characterized by enzyme loss from cells (creatine kinase, lactate dehydrogenase). Cardiomyocytes reoxygenated after 120 min hypoxia hypercontracted, but enhanced enzyme loss was only observed at 80 mOsm. The NO donors SIN-1 (10 mM), sodium nitroprusside (10 mM), S-nitroso-N-acetyl-D,L -penicillamine (SNAP, 100 [mu]M) and the anti-lipid peroxidant diphenylphenylenediamine (DPPD, 2.5 [mu]M) reduced enzyme loss upon hypoosmolal reoxygenation. Agents activating cyclic-GMP dependent pathways (atrionatriuretic peptide (1 [mu]M), urodilatin (1 [mu]M), and 8-bromo-cyclo-GMP (10 mM)), the contractile inhibitor 2,3 -butanedione monoxime (10 mM) and the SIN-1 metabolite SIN-1C (10 mM) did not protect cardiomyocytes against osmotic fragility. The results show that increased osmotic fragility of isolated adult rat cardiomyocytes can be prevented at the time of reoxygenation by NO donors and DPPD, in a cyclic-GMP independent way.

Received 24 February 1995; accepted in final form 17 January
1996.
APS Manuscript Number H176-5.
Article publication pending Am. J. Physiol. (Heart Circ. Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 8 February 96