Evidence for cgmp mediation of skeletal muscle arteriolar dilation to lactate. Chen, Ya-Li, Michael S. Wolin, and Edward J. Messina. Department of Physiology, New York Medical College, Valhalla, New York 10595
APStracts 3:0118A, 1996.
In this study we tested the hypothesis that lactate, independent of changes in pH, can effect skeletal muscle blood flow through arteriolar dilation that may be mediated by cGMP. Isolated, cannulated and pressurized first order rat cremaster skeletal muscle arterioles were studied in a myograph chamber containing Krebs bicarbonate buffer under no-flow conditions. At pH 7.4 and a PO2 of 65 mmHg, neutralized lactic acid (lactate) and pyruvic acid (pyruvate) caused arteriolar dilation over the 1-10 mM concentration range. This response to lactate was not altered by 10-5 M indomethacin (IND), 10-4 M nitro-L-arginine (L-NNA) or by removal of the endothelium. However, responses to 1, and 3 mM pyruvate were significantly inhibited 100% by endothelium removal and that to 10mM 71%. The relaxation of endothelium denuded arterioles to lactate was inhibited by 10 [mu]M methylene blue (MB), or 10 [mu]M LY83583, and by hypoxia (PO2 = 7-10 mmHg) or diphenyliodonium, an inhibitor of superoxide producing flavoprotein enzymes. In contrast, arteriolar dilation to the acidification of the Krebs buffer to pH 7.15, produced by increasing the CO2 concentration of the gas mixture from 5% to 10%, was not inhibited by MB. These results are consistent with lactate induced skeletal muscle arteriolar dilation being dependent upon H2O2 mediated activation of vascular smooth muscle guanylate cyclase and independent of endothelium-derived mediators.

Received 28 September 1995; accepted in final form 6 February
1996.
APS Manuscript Number A1048-5.
Article publication pending Journal of Applied Physiology.
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 13 March 96