Leptin increases energy expenditure and selectively promotes fat metabolism in ob/ob mice. Hwa, Joyce J., Ahmad B. Fawzi, Michael P. Graziano, Lorraine Ghibaudi, Patricia Williams, Margaret Van Heek, Harry Davis, Mark Rudinski, Edmund Sybertz, and Catherine D. Strader. Department of CNS and Cardiovascular Research, Schering-Plough Research Institute, Kenilworth, New Jersey 07033
APStracts 3:0421R, 1996.
Obesity occurs whenever energy intake exceeds energy expenditure. The ob gene product, leptin, is a potent anorectic agent when administered to ob/ob mice, but its effects on energy expenditure have not been investigated in detail. The present study was designed to analyze the acute metabolic effects of leptin in vivo. Analysis of oxygen consumption in ob/ob mice demonstrated a reduction in energy expenditure compared to lean controls; this reduction showed a diurnal fluctuation and was most evident during the light cycle. A single intraperitoneal dose of leptin increased oxygen consumption during the light cycle in ob/ob mice, ablating the circadian fluctuation in this parameter. In addition, leptin had a profound effect on fuel selection: the respiratory quotient was markedly reduced, indicating a reduction in carbohydrate oxidation and an increase in fat oxidation. These acute effects of leptin on metabolic parameters are consistent with the selective loss of body fat observed upon chronic leptin treatment and suggest that increased energy utilization plays an important role in the anti-obese actions of leptin.

Received 8 August 1996; accepted in final form 5 November 1996.
APS Manuscript Number R468-6.
Article publication pending Am. J. Physiol. (Regulatory Integrative
Comp. Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 31 December 1996