Functional evidence for l-type ca2+ channels controlling adrenal catecholamine release induced by angiotensin ii in vivo. Martineau, Daniel, Richard Briand, and Nobuharu Yamaguchi. Groupe de recherche sur le syst[grave]eme nerveux autonome, Facult[acute]e de pharmacie, Universit[acute]e de Montr[acute]eal, C.P. 6128, Centreville, Montr[acute]eal, QC, H3C 3J7, Canada, Bristol-Myers Squibb (Canada), 2365 ch. C[circumflex]ote-de-Liesse, Montr[acute]eal, QC, H4N 2M7, Canada
APStracts 3:0234R, 1996.
The aim of the present study was to investigate the functional involvement of L- and/or N-type Ca2+ channels in adrenal catecholamine secretion in response to exogenous angiotensin II in anesthetized dogs. Plasma catecholamine concentrations in adrenal venous and aortic blood were determined by an HPLC-electrochemical method. In the first series of experiments, repeated infusions of BAY-K 8644 locally administered into the left adrenal gland with an interval of 15 min resulted in significant and reproducible increases in adrenal catecholamine secretion. Nifedipine, similarly administered 5 min prior to BAY-K 8644, diminished BAY-K 8644-induced catecholamine secretion in a dose-dependent manner and completely blocked the catecholamine response with the highest dose tested. In the second series, locally infused angiotensin II resulted in a significant increase in adrenal catecholamine secretion. The maximum catecholamine response to angiotensin II was attenuated by approximately 65% in the presence of nifedipine with the dose that abolished the BAY-K 8644-induced catecholamine release. This inhibition by nifedipine remained unchanged in the presence of additional -conotoxin. The present study shows that dihydropyridine -sensitive L-type Ca2+ channels are operative in the adrenal medulla of the dog in vivo. The results indicate that the L-type Ca2+ channels are only partially implicated in the local regulation of angiotensin II-induced adrenal catecholamine secretion, suggesting the existence of another mechanism. However, -conotoxin-sensitive N -type Ca2+ channels are unlikely to be functionally involved in postsynaptic mechanisms mediating adrenal catecholamine secretion in response to exogenous angiotensin II under in vivo conditions.

Received 28 September 1995; accepted in final form 30 May 1996.
APS Manuscript Number R609-5.
Article publication pending Am. J. Physiol. (Regulatory Integrative
Comp. Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 4 July 96