Rapid redistribution and inhibition of renal sodium transporters during natriuresis induced by acute hypertension. Zhang, Yibin, Austin K. Mircheff, Charles B. Hensley, Clara E. Magyar, David G. Warnock, Regine Chambrey, Kay-Pong Yip, Donald J. Marsh, Niels-H. Holstein Rathlou, and Alicia A. McDonough. Department of Physiology and Biophysics, University of Southern California School of Medicine, Departments of Medicine and Physiology and Biophysics, Nephrology Research and Training Center, Vascular Biology and Hypertension Program, University of Alabama at Birmingham and Department of Veterans Affairs, Department of Physiology, Brown University School of Medicine, and University Institute of Experimental Medicine, Panum Institute, Copenhagen, Denmark
APStracts 3:0023F, 1996.
Acute arterial hypertension provokes a rapid decrease in proximal tubule sodium reabsorption, increasing flow to the macula densa, the signal for tubuloglomerular feedback. We tested the hypothesis, in rats, that sodium transport is decreased due to rapid redistribution of apical Na/H exchangers and basolateral sodium pumps to internal membranes. Arterial pressure was increased 50 mm by constricting various arteries. We also tested whether transporter internalization occurred when proximal tubule sodium reabsorption was inhibited with the carbonic anhydrase inhibitor benzolamide. Five min after initiating either natriuretic stimuli, cortex was removed and membranes fractionated by density gradient centrifugation. Urine output and endogenous lithium clearance increased 3 fold in response to either stimuli. Acute hypertension provoked a redistribution of apical NHE-3, alkaline phosphatase and dipeptidyl peptidase IV to higher density membranes enriched in the intracellular membrane markers. Basolateral membrane Na,K-ATPase activity decreased 50%, 25 -30% of the [alpha]1 and [beta]1 subunits redistributed to higher density membranes, and the remainder is attributed to decreased activity of the transporters. Benzolamide did not alter sodium transporter activity or distribution, implying that decreasing apical Na+ uptake does not initiate redistribution or inhibition of basolateral Na,K-ATPase. We conclude that proximal tubule natriuresis provoked by acute arterial pressure is mediated by both endocytic removal of apical Na/H exchangers and basolateral sodium pumps as well as decreased total sodium pump activity.

Received 31 July 1995; accepted in final form 25 January 1996.
APS Manuscript Number F250-5.
Article publication pending Am. J. Physiol. (Renal Fluid Electrolyte
Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 8 February 96