Direct demonstration of aquaporin-2 water channel recycling in stably transfected llc-pk1 epithelial cells. Katsura, Toshiya, Dennis A. Ausiello, and Dennis Brown. Renal Unit, Massachusetts General Hospital and Departments of Medicine and Pathology, Harvard Medical School, Boston, Massachusetts 02114
APStracts 3:0010F, 1996.
Vasopressin dependent membrane insertion of aquaporin-2 (AQP2) in collecting duct principal cells has been demonstrated in vivo and in vitro. However, the hypothesis that the AQP2 molecule recycles between intracellular vesicles and the plasma membrane in response to hormonal stimulation and withdrawal remains to be demonstrated directly. In the present study, we examined AQP2 recycling between intracellular vesicles and the plasma membrane in the absence of de novo protein synthesis using LLC-PK1 cells transfected with an AQP2 -c-myc construct. Cells were treated with cycloheximide for 30 min prior to vasopressin stimulation and all subsequent treatments were performed in the continued presence of cycloheximide. Complete inhibition of AQP2 biosynthesis by cycloheximide was verified by immunoprecipitation. Immunofluorescence revealed that AQP2 was located on intracellular vesicles in non-stimulated cells, but was relocated to the plasma membrane after vasopressin treatment even in the presence of cycloheximide. After vasopressin washout AQP2 was retrieved to intracellular vesicles, and was relocated to the plasma membrane after restimulation with forskolin. Subsequent forskolin washout resulted in AQP2 endocytosis, and a second stimulation with forskolin resulted in relocation to the plasma membrane. These data, obtained in the absence of de novo protein synthesis, clearly indicate that AQP2 can be recycled multiple times between intracellular vesicles and the plasma membrane.

Received 6 September 1995; accepted in final form 18 December
1995.
APS Manuscript Number F295-5.
Article publication pending Am. J. Physiol. (Renal Fluid Electrolyte
Physiology).
ISSN 1080-4757 Copyright 1996 The American Physiological Society.
Published in APStracts on 22 January 96