Progesterone-induced changes in sleep in male subjects. Friess, Elisabeth, Hirokuni Tagaya, Lorenz Trachsel, Florian Holsboer, and Rainer Rupprecht. Max Planck Institute of Psychiatry, Clinical Institute, Department of Psychiatry, D-80804 Munich, Germany
APStracts 4:0012E, 1997.
Progesterone administration induces a reduction of the vigilance state in humans during wakefulness. It has been been suggested that this effect is mediated via neuroactive metabolites that interact with the -aminobutyric acid (GABAA) receptor complex. To investigate the effects of progesterone administration on the sleep electroencephalogram (EEG) in humans we made polysomnographic recordings, including sleep-stage specific spectral analysis, and concomitantly measured plasma concentrations of progesterone and its GABA-active metabolites 3[alpha]-hydroxy-5[alpha]-dihydroprogesterone (allopregnanolone) and 3[alpha]-hydroxy-5[beta]-dihydroprogesterone (pregnanolone) in 9 healthy male subjects in a double-blind placebo -controlled cross-over study. Progesterone administration at 9:30 p.m. induced a significant increase in the amount of non-REM sleep. The EEG spectral power during non-REM sleep showed a significant decrease in the slow wave frequency range (0.4-4.3 Hz), whereas the spectral power in the higher frequency range (>15 Hz) tended to be elevated. Some of the observed changes in sleep architecture and sleep-EEG power spectra are similar to those induced by agonistic modulators of the GABAA receptor complex and appear to be mediated in part via the conversion of progesterone into its GABA-active metabolites.

Received 27 April 1996; accepted in final form 6 January 1997.
APS Manuscript Number E485-6.
Article publication pending Am. J. Physiol. (Endocrinol. Metab.).
ISSN 1080-4757 Copyright 1997 The American Physiological Society.
Published in APStracts on 19 February 1997