Sodium-gated cation channel implicated in the activation of lobster olfactory receptor neurons. Aslbek B. Zhainazarov, Richard E. Doolin, and Barry W. Ache.. Whitney Laboratory and Depts. of Zoology and Neuroscience, Univ. of Florida, St. Augustine, FL 32086-8623..
APStracts 4:315N, 1997.
ABSTRACT
The role of Na+-activated channels in cellular function, if any, is still elusive. Here, we implicate a Na+-activated nonselective cation channel in the activation of lobster olfactory receptor neurons. We show that a Na+-activated channel occurs in the transduction compartment (outer dendrite) of the receptor cells. The channel density in the outer dendrite (17.3 æm-2) is two orders of magnitude greater than that in the soma of the cells (0.06 æm-2). The properties of the channel in the outer dendrite are identical to those described earlier in detail for a Na+-activated channel on the soma of the cells in culture. The channel is specifically activated by intracellular Na+ in a concentration-dependent manner [EC50= 49.2ñ3.0 (S.E.M.) mM] in cell-free patches in the absence of both divalent cations and nucleoside triphosphates. The presence of a Na+-activated channel in a cellular compartment specialized for odor transduction suggests that the channel functions in odor activation. Two separate lines of experimental evidence support this view. (1) Two pharmacological probes (W7 and trifluoperazine) which block the Na+-gated channel from outside in excised patches [IC50: 16.3ñ1.5 (S.E.M.) æM for W7; 14.4ñ0.9 æM for trifluoperazine], significantly reduce odor-evoked responses when applied focally to the outer dendrite of the cells. (2) The response of the cells to odors is specific for Na+. Substituting Na+ with either Li+ or NH4+, both of which permeate the cell but do not activate the Na+-gated channel, also significantly reduces the odor-evoked response of the cells, implying that a substantial part of the odor-evoked depolarization can be ascribed to a Na+-activated conductance. We hypothesize, therefore, that the Na+-activated channel amplifies the receptor current as a result of being secondarily activated by the primary odor transduction pathway.

Received 18 September 1997; accepted in final form 4 November 1997.
APS Manuscript Number J769-7.
Article publication pending J. Neurophysiol.
ISSN 1080-4757 Copyright 1997 The American Physiological Society.
Published in APStracts on 14 November 1997